Gallamine is an allosteric, selective muscarinic M2 acetylcholine receptor antagonist (EC50: 130 nM for [3H]NMS dissociation from porcine muscarinic M2 receptors). Gallamine is also an acetylcholinesterase inhibitor (IC50s : 1070 µM, 1480 µM, 235 µM for EeAChE, hAChE, hBChE, respectively (in the absence of MeCN)). Gallamine increases free norepinephrine levels. Gallamine can be used as a muscle relaxant[1][2].
Molekulargewicht:
423.63
CAS Nummer:
[153-76-4]
Formel:
C24H45N3O3
Target-Kategorie:
Cholinesterase (ChE),mAChR
Anwendungsbeschreibung:
MCE Product type: Reference compound1
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