NEP108 is a GID4 E3 ligase-based BRD4 PROTAC degrader, with its DC50 value approximately 3.8 µM. NEP108 has a strong affinity for GID4, with a KD value of 0.22 µM, and the KD value of its trimeric complex is 2.85 µM. NEP108 can be used for cancer research[1].
Molekulargewicht:
887.49
CAS Nummer:
[3031840-31-7]
Formel:
C47H51ClN10O4S
Target-Kategorie:
Epigenetic Reader Domain,PROTACs
Anwendungsbeschreibung:
MCE Product type: Reference compound
* Mehrwertsteuer und Versandkosten nicht enthalten. Irrtümer und Preisänderungen vorbehalten