S1RA (hydrochloride), CAS [[1265917-14-3]]

Produktübersicht

• Artikelname: S1RA (hydrochloride), CAS [[1265917-14-3]]
• Artikelnummer: MCE-HY-18099A
• Hersteller Artikelnummer: HY-18099A
• Alternativnummer: MCE-HY-18099A-10MMX1ML,MCE-HY-18099A-5MG,MCE-HY-18099A-100MG,MCE-HY-18099A-10MG,MCE-HY-18099A-50MG,MCE-HY-18099A-25MG,MCE-HY-18099A-250MG
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien
• Alternative Synonym: E-52862 hydrochloride

Produktbeschreibung

S1RA (E-52862) hydrochloride is an orally active and selective sigma-1 receptor (sigma1R) antagonist with a Ki value of 17 nM. S1RA hydrochloride shows good selectivity against sigma2R (Ki >1000 nM). S1RA hydrochloride is a human 5-HT2B receptor antagonist with an IC50 value of 4.7 µM. S1RA hydrochloride inhibits neuropathic pain and activity-induced spinal sensitization[1][2].

Produkteigenschaften

• Molekulargewicht: 373.88
• Reinheit: 99.94
• CAS Nummer: [1265917-14-3]
• Formel: C20H24ClN3O2
• Target-Kategorie: 5-HT Receptor,Sigma Receptor

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound