CBX2-IN-1 is a CBX2 inhibitor with an IC50 of 9.6 µM. CBX2-IN-1 binds the CBX2 chromodomains H3K27me3 binding channel, blocks interaction between CBX2 and H3K27me3, and exhibits selective affinity toward CBX2, CBX4, CBX6, CBX7, and CBX8 over CBX1, CBX3, and CBX5. CBX2-IN-1 can be used for the research of prostate cancers[1].
Molekulargewicht:
465.54
Formel:
C29H27N3O3
Target-Kategorie:
Histone Methyltransferase
Anwendungsbeschreibung:
MCE Product type: Reference compound
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