GPX4 degrader-1, CAS [[3057531-85-5]] Preis auf Anfrage
Artikelnummer:
MCE-HY-181598
| Artikelname: |
GPX4 degrader-1, CAS [[3057531-85-5]] Preis auf Anfrage |
| Artikelnummer: |
MCE-HY-181598 |
| Hersteller Artikelnummer: |
HY-181598 |
| Alternativnummer: |
MCE-HY-181598-1UNIT |
| Hersteller: |
MedchemExpress |
| Kategorie: |
Biochemikalien |
| GPX4 degrader-1 (Compound RS-1) is a hydrophobic tagging (HyT)-mediated GPX4 degrader (DC50: 8.9 nM in HT1080 cells) GPX4 degrader-1 induces GPX4 degradation. GPX4 degrader-1 induces Ferroptosis. GPX4 degrader-1 increases lipid ROS. GPX4 degrader-1 demonstrates potent antitumor efficacy in a murine mammary carcinoma model[1]. |
| Molekulargewicht: |
634.16 |
| CAS Nummer: |
[3057531-85-5] |
| Formel: |
C38H36ClN3O4 |
| Target-Kategorie: |
Ferroptosis,Glutathione Peroxidase,Reactive Oxygen Species (ROS) |
| Anwendungsbeschreibung: |
MCE Product type: Reference compound |