SM-11044 is a beta-adrenoceptor agonist with Ki values of 18.1 µM (beta1), 4.1 µM (beta2) and 1.3 µM (beta3), showing higher binding selectivity for the beta3-adrenoceptor. SM-11044 stimulates cAMP accumulation in cells expressing this receptor. SM-11044 mediates ileal relaxation, tracheal relaxation, pulmonary parenchymal relaxation, increased right atrial heart rate and adipocyte lipolysis[1].
Molekulargewicht:
483.37
CAS Nummer:
[142784-65-4]
Formel:
C22H28BrFN2O4
Target-Kategorie:
Adrenergic Receptor
Anwendungsbeschreibung:
MCE Product type: Reference compound
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