JNK1 degrader-1 is a JNK1 HyT degrader. JNK1 degrader-1 can induce JNK1 degradation through the HyT-mediated ubiquitin-proteasome system and autophagy-lysosome pathway. JNK1 degrader-1 inhibits TGF-beta1-induced epithelial-mesenchymal transition (EMT). JNK1 degrader-1 can be used for research on fibrotic diseases and cancer metastasis. (Pink: JNK1 ligand (HY-183006), Blue: Hyt hydrophobic group (HY-W037848), Black: Linker (HY-B1008))[1].
Molekulargewicht:
575.50
Formel:
C29H31BrN6O2
Target-Kategorie:
HyT,JNK
Anwendungsbeschreibung:
MCE Product type: Reference compound
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