SSTR5/TGR5-modulator-1, CAS [[3069267-46-2]] Preis auf Anfrage

Produktübersicht

• Artikelname: SSTR5/TGR5-modulator-1, CAS [[3069267-46-2]] Preis auf Anfrage
• Artikelnummer: MCE-HY-182905
• Hersteller Artikelnummer: HY-182905
• Alternativnummer: MCE-HY-182905-1UNIT
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien

Produktbeschreibung

SSTR5/TGR5-modulator-1 is an orally active and dual-target small molecule, balanced in vitro activity at human TGR5 and human SSTR5. SSTR5/TGR5-modulator-1 activates human TGR5 to promote cAMP accumulation. SSTR5/TGR5-modulator-1 blocks human SSTR5 to inhibit agonist-induced calcium mobilization. SSTR5/TGR5-modulator-1 improves glucose tolerance in mice. SSTR5/TGR5-modulator-1 alleviates gallbladder filling in mice at pharmacologically relevant doses. SSTR5/TGR5-modulator-1 has suboptimal physicochemical and metabolic properties.SSTR5/TGR5-modulator-1 can be used for the research of type 2 diabetes mellitus[1].

Produkteigenschaften

• Molekulargewicht: 727.87
• CAS Nummer: [3069267-46-2]
• Formel: C39H45N5O7S
• Target-Kategorie: G protein-coupled Bile Acid Receptor 1,Somatostatin Receptor

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound