Emixustat is an orally active RPE65 inhibitor with an IC50 value of 4.4 nM. Emixustat is also a visual cycle modulator, capable of regulating visual cycle activity by inhibiting retinol isomerization, and holds potential for studying vision disorders such as age-related macular degeneration (AMD)[1][2][3][4].
Molekulargewicht:
263.38
Reinheit:
98.74
CAS Nummer:
[1141777-14-1]
Formel:
C16H25NO2
Target-Kategorie:
RPE65
Anwendungsbeschreibung:
Reference compound
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