Avitinib (maleate), CAS [[1557268-88-8]]

Artikelnummer: MCE-HY-19816A
Artikelname: Avitinib (maleate), CAS [[1557268-88-8]]
Artikelnummer: MCE-HY-19816A
Hersteller Artikelnummer: HY-19816A
Alternativnummer: MCE-HY-19816A-5MG,MCE-HY-19816A-10MG,MCE-HY-19816A-50MG,MCE-HY-19816A-100MG,MCE-HY-19816A-25MG,MCE-HY-19816A-10MMX1ML
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Alternative Synonym: Abivertinib (maleate), AC0010 (maleate)
Avitinib (Abivertinib) maleate is a third-generation, irreversible and orally active selective EGFR inhibitor, with IC50 values of 0.18 nM, 0.18 nM, 7.68 nM and against EGFR L858R, EGFR T790M and wild-type EGFR. Avitinib maleate is also a BTK inhibitor that induces apoptosis and inhibits phosphorylation of BTK in mantle cell lymphoma. Avitinib maleate shows anticancer effects[1][2].
Molekulargewicht: 603.60
Reinheit: 99.86
CAS Nummer: [1557268-88-8]
Formel: C30H30FN7O6
Target-Kategorie: Apoptosis,Btk,EGFR
Anwendungsbeschreibung: MCE Product type: Reference compound