Ruxolitinib-d9, CAS [[1513883-55-0]] Preis auf Anfrage
Artikelnummer:
MCE-HY-50856S2
Hersteller Artikelnummer:
HY-50856S2
Alternativnummer:
MCE-HY-50856S2-1UNIT
Hersteller:
MedchemExpress
Kategorie:
Biochemikalien
Alternative Synonym:
INCB18424-d9
Ruxolitinib-d9 (INCB18424-d9) is deuterium labeled Ruxolitinib. Ruxolitinib (INCB18424) is an orally active and selective JAK1/2 inhibitor with IC50s of 3.3 nM and 2.8 nM in cell-free assays, and has 130-fold selectivity for JAK1/2 over JAK3[1]. Ruxolitinib induces autophagy and kills tumor cells through toxic mitophagy[3].