Safinamide (Standard), CAS [[133865-89-1]] Preis auf Anfrage

Artikelnummer: MCE-HY-70057R
Artikelname: Safinamide (Standard), CAS [[133865-89-1]] Preis auf Anfrage
Artikelnummer: MCE-HY-70057R
Hersteller Artikelnummer: HY-70057R
Alternativnummer: MCE-HY-70057R-100MG,MCE-HY-70057R-5MG,MCE-HY-70057R-25MG,MCE-HY-70057R-50MG,MCE-HY-70057R-10MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Alternative Synonym: FCE 26743 (Standard), EMD 1195686 (Standard)
Safinamide (Standard) is the analytical standard of Safinamide. This product is intended for research and analytical applications. Safinamide is a potent, selective, and reversible monoamine oxidase B (MAO-B) inhibitor (IC50=0.098 µM) over MAO-A (IC50=580 µM)[1]. Safinamide also blocks sodium channels and modulates glutamate (Glu) release, showing a greater affinity at depolarized (IC50=8 µM) than at resting (IC50=262 µM) potentials. Safinamide has neuroprotective and neurorescuing effects and can be used for the study of parkinson disease, ischemia stroke etc.al[2][3].
Molekulargewicht: 302.34
CAS Nummer: [133865-89-1]
Formel: C17H19FN2O2
Target-Kategorie: Monoamine Oxidase,Reference Standards
Anwendungsbeschreibung: MCE Product type: Reference Standards