Ropivacaine-d7 (hydrochloride), CAS [[1217667-10-1]]
Artikelnummer:
MCE-HY-B0563BS
Hersteller Artikelnummer:
HY-B0563BS
Alternativnummer:
MCE-HY-B0563BS-1MG
Hersteller:
MedchemExpress
Kategorie:
Biochemikalien
Ropivacaine-d7 hydrochloride is a deuterium labeled Ropivacaine (hydrochloride) (HY-B0563B)[1]. Ropivacaine hydrochloride is a potent sodium channel blocker and blocks impulse conduction via reversible inhibition of sodium ion influx in nerve fibrese[2][3]. Ropivacaine is also an inhibitor of K2P (two-pore domain potassium channel) TREK-1 with an IC50 of 402.7 µM in COS-7 cells membrane[4]. Ropivacaine is widely used for neuropathic pain management in vivo[2].