Desvenlafaxine succinate hydrate, the succinate salt form of the isolated major active metabolite of Venlafaxine (HY-B0196), is an orally active and BBB penetrated 5-HT and norepinephrine reuptake inhibitor, with IC50 values of 47.3 nM and 531.3 nM for hSERT and hNET, respectively. Desvenlafaxine succinate hydrate shows weak binding affinity (62% inhibition at 100 µM) at the human dopamine (DA) transporter[1][2].
Molekulargewicht:
399.48
Reinheit:
99.82
CAS Nummer:
[386750-22-7]
Formel:
C20H33NO7
Target-Kategorie:
Serotonin Transporter
Anwendungsbeschreibung:
MCE Product type: Reference compound
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