Telenzepine is an antimuscarinic agent with Kis of 0.94 nM (M1 mAChR) and 17.8 nM (M2 mAChR) binding to muscarinic receptors. Telenzepine effectively blocks synaptic transmission promoted by muscarinic or M1 receptor agonists. Thus, Telenzepine can reduce the amplitude of extracellular slow excitatory postsynaptic potentials (EC50=38 nM) and slow inhibitory postsynaptic potentials (EC50=253 nM)[1].
Molekulargewicht:
370.47
CAS Nummer:
[80880-90-6]
Formel:
C19H22N4O2S
Target-Kategorie:
mAChR
Anwendungsbeschreibung:
MCE Product type: Reference compound
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