Nonapeptide-1 (Melanostatine-5) acetate salt, a peptide hormone, is a selective antagonist of MC1R (Ki: 40 nM). Nonapeptide-1 acetate salt is a competitive alpha-MSH antagonist that potently inhibits intracellular cAMP and melanosome dispersion induced by alpha-MSH in melanocytes (IC50: 2.5 nM and 11 nM, respectively). Nonapeptide-1 acetate salt inhibits melanin synthesis, and can be used in the research of skin pigmentation and regulation of steroid production in the adrenal gland, skin cancer[1][2][3].
Molekulargewicht:
1266.56
Reinheit:
95.58
Formel:
C63H91N15O11S
Target-Kategorie:
Melanocortin Receptor
Anwendungsbeschreibung:
Peptides
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