PSMA-D5 has a binding affinity for PSMA with Ki of 0.21 nM and can be used for PSMA tracing after radiolabeling. PSMA-D5 ([68Ga]-labeled) contains a DOTA chelator, allowing convenient labeling with therapeutic radionuclides such as 177Lu and 225Ac. PSMA-D5 ([68Ga]-labeled) shows excellent pharmacokinetic properties, exhibiting remarkable tumor uptake in 22Rv1 tumors[1]. PSMA-D5 can be used for the synthesis/research of Radionuclide-Drug Conjugates (RDCs).
Molekulargewicht:
1317.31
Reinheit:
98.61
CAS Nummer:
[3056440-83-3]
Formel:
C57H80N12O24
Target-Kategorie:
PSMA,Radionuclide-Drug Conjugates (RDCs)
Anwendungsbeschreibung:
Peptides
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