Phrixotoxin 3-NH2 (TFA)

Produktübersicht

• Artikelname: Phrixotoxin 3-NH2 (TFA)
• Artikelnummer: MCE-HY-P1218B
• Hersteller Artikelnummer: HY-P1218B
• Alternativnummer: MCE-HY-P1218B-500UG,MCE-HY-P1218B-100UG,MCE-HY-P1218B-1MG
• Hersteller: MedchemExpress
• Kategorie: Proteine/Peptide

Produktbeschreibung

Phrixotoxin 3-NH2 TFA is a derivative of Phrixotoxin 3 TFA (HY-P1218A). Phrixotoxin 3 TFA is a potent blocker of voltage-gated sodium channels, with IC50s of 0.6, 42, 72, 288, 610 nM for NaV1.2, NaV1.3, NaV1.4, NaV1.1 and NaV1.5, respectively. Phrixotoxin 3 TFA modulates voltage-gated sodium channels with properties similar to those of typical gating-modifier toxins, both by causing a depolarizing shift in gating kinetics and by blocking the inward component of the sodium current[1].

Produkteigenschaften

• Molekulargewicht: 4058.74 (free base)
• Reinheit: 98.96
• Formel: C176H270N52O47S6.xC2HF3O2
• Target-Kategorie: Sodium Channel

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Peptides