[DArg10, DAla20] TLQP-21, TLQP-21 (HY-P1345) analogue, is a C3aR agonist (EC50: 87 nM for beta-arrestin recruitment). [DArg10, DAla20] TLQP-21 elicits calcium influx. [DArg10, DAla20] TLQP-21 slightly but not significantly potentiates adrenergic-induced lipolysis. [DArg10, DAla20] TLQP-21 can be used in the research of inflammatory diseases, metabolic disorders, and neurological conditions[1].
Molekulargewicht:
2432.75
Formel:
C107H170N40O26
Target-Kategorie:
Calcium Channel,Complement System,Drug Derivative
Anwendungsbeschreibung:
MCE Product type: Peptides
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