L-771688 (hydrochloride), CAS [[200051-19-0]] Preis auf Anfrage

Produktübersicht

• Artikelname: L-771688 (hydrochloride), CAS [[200051-19-0]] Preis auf Anfrage
• Artikelnummer: MCE-HY-U00237B
• Hersteller Artikelnummer: HY-U00237B
• Alternativnummer: MCE-HY-U00237B-1UNIT
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien

Produktbeschreibung

L-771688 hydrochloride is a potent and highly selective alpha1A-adrenoceptor antagonist (Kd=43-90 pM). L-771688 hydrochloride is effective against cloned human, rat and dog alpha1A-adrenergic receptors. L-771688 exhibits high affinity (Ki 1 nM) and over 500-fold selectivity over the alpha1B and alpha1D isoforms. L-771688 potently antagonizes norepinephrine-induced responses at these receptors. Inhibits contractions induced by phenylephrine or A-61603 in rat, dog, human and monkey models[1].

Produkteigenschaften

• Molekulargewicht: 630.51
• CAS Nummer: [200051-19-0]
• Formel: C28H35Cl2F2N5O5
• Target-Kategorie: Adrenergic Receptor

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound