WX2-43, CAS [[723754-14-1]]

Artikelnummer: MCE-HY-W072962
Artikelname: WX2-43, CAS [[723754-14-1]]
Artikelnummer: MCE-HY-W072962
Hersteller Artikelnummer: HY-W072962
Alternativnummer: MCE-HY-W072962-10MMX1ML,MCE-HY-W072962-100MG,MCE-HY-W072962-5MG,MCE-HY-W072962-10MG,MCE-HY-W072962-25MG,MCE-HY-W072962-50MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
WX2-43 is a PRMT5-KLF4 inhibitor (Kd of 11.0 nM). WX2-43 binds to the region between amino acids L400-M500 on PRMT5. WX2-43 efficiently intercepts the interaction between KLF4 and PRMT5, and blocks KLF4 methylation. WX2-43 decreases p21 levels and increases Bax levels. WX2-43 suppresses triple negative breast tumor progression. WX2-43 can be used in the research of triple-negative breast cancer and colorectal cancer[1][2].
Molekulargewicht: 288.82
Reinheit: 98.74
CAS Nummer: [723754-14-1]
Formel: C17H21ClN2
Target-Kategorie: Bcl-2 Family,Histone Methyltransferase,KLF,PAK
Anwendungsbeschreibung: MCE Product type: Reference compound