ID110460002, CAS [[1172882-21-1]] Preis auf Anfrage
Artikelnummer:
MCE-HY-W414109
Hersteller Artikelnummer:
HY-W414109
Alternativnummer:
MCE-HY-W414109-1UNIT
Hersteller:
MedchemExpress
Kategorie:
Biochemikalien
ID110460002 possesses both full agonist activity at the µ-opioid receptor (OPRM) and agonist activity at the delta-opioid receptor (OPRD). ID110460002 acts as a potent agonist for the G protein pathways of both receptors, but exhibits only very weak partial agonist activity towards the beta-arrestin-2 pathway. The agonistic potency of ID110460002 at OPRM has extremely high intrinsic activity and is unaffected by reduced receptor expression levels, while its potency at OPRD depends on receptor expression levels. ID110460002 displays tissue- or organ-dependent properties, and serves as a critical compound for investigating pain mechanisms and analgesia[1].
Molekulargewicht:
356.45
CAS Nummer:
[1172882-21-1]
Formel:
C20H25FN4O
Target-Kategorie:
Arrestin,Opioid Receptor
Anwendungsbeschreibung:
MCE Product type: Reference compound
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