Samuraciclib hydrochloride, CAS [[1805789-54-1]]

Artikelnummer: TGM-T10898
Artikelname: Samuraciclib hydrochloride, CAS [[1805789-54-1]]
Artikelnummer: TGM-T10898
Hersteller Artikelnummer: T10898
Alternativnummer: TGM-T10898-1MLX10MM(INDMSO),TGM-T10898-1MG,TGM-T10898-2MG,TGM-T10898-5MG,TGM-T10898-10MG,TGM-T10898-25MG,TGM-T10898-50MG,TGM-T10898-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
Alternative Synonym: ICEC0942 hydrochloride , CT7001 hydrochloride
Samuraciclib hydrochloride (ICEC0942 hydrochloride) is a potent, selective, ATP competitive and oral active CDK7 inhibitor with IC50 of 41 nM. The selectivity of Samuraciclib hydrochloride is 45-, 15-, 230- and 30-fold higher than CDK1, CDK2 (IC50 is 578 nM), CDK5 and CDK9 respectively. Samuraciclib hydrochloride inhibits the growth of breast cancer cell lines with GI50 values between 0.2-0.3 µM. Samuraciclib hydrochloride has anti-tumor effects.
Molekulargewicht: 430.97
Reinheit: 0.998
CAS Nummer: [1805789-54-1]
Formel: C22H31ClN6O
Target-Kategorie: Apoptosis|||CDK
T10898