Heptamidine dimethanesulfonate (SBi4211 dimethanesulfonate) serves as a potent inhibitor related to Pentamidine, targeting the calcium-binding protein S100B with a dissociation constant (Kd) of 6.9 µM. It demonstrates specificity by preferentially killing melanoma cells overexpressing S100B compared to cells lacking this protein. Additionally, Heptamidine is employed as a valuable research tool in the study of Myotonic dystrophy (DM).
Molekulargewicht:
560.68
Reinheit:
97.80%
CAS Nummer:
[161374-55-6]
Formel:
C23H36N4O8S2
Target-Kategorie:
Others
T11553
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