JTV-519 free base (K201 free base), known for its antiarrhythmic and cardioprotective properties, acts as a Ca2+-dependent blocker of sarcoplasmic reticulum Ca2+-stimulated ATPase (SERCA) and as a partial agonist of ryanodine receptors in striated muscle.
Molekulargewicht:
424.6
CAS Nummer:
[145903-06-6]
Formel:
C25H32N2O2S
Target-Kategorie:
Calcium Channel|||FLT
T11731
T11731
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