CLP257, CAS [[1181081-71-9]]

Artikelnummer: TGM-T14984
Artikelname: CLP257, CAS [[1181081-71-9]]
Artikelnummer: TGM-T14984
Hersteller Artikelnummer: T14984
Alternativnummer: TGM-T14984-1MG,TGM-T14984-2MG,TGM-T14984-5MG,TGM-T14984-10MG,TGM-T14984-25MG,TGM-T14984-50MG,TGM-T14984-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
CLP257 is a selective K+-Cl- cotransporter KCC2 activator (EC50: 616 nM) and it is inactive against NKCC1, GABAA receptors, KCC1, KCC3 or KCC4. CLP257 alleviates hypersensitivity in rats with neuropathic painc and it also modulates plasmalemmal KCC2 protein turnover post-translationally. CLP257 restores impaired Cl- transport in neurons with diminished KCC2 activity.
Molekulargewicht: 307.34
Reinheit: 98.13%
CAS Nummer: [1181081-71-9]
Formel: C14H14FN3O2S
Target-Kategorie: Potassium Channel
T14984