Didesmethyl cariprazine, a metabolite of Cariprazine, is the major cyclic active part. Didesmethyl cariprazine has a long half-life of 1-3 weeks. Cariprazine is a potent D3 preference D3/D2 receptor partial agonist of dopamine for the treatment of schizophrenia, bipolar mania, and depression, with a high affinity for d3 and d2 receptors and a moderate affinity for 5-HT 1A receptors.
Molekulargewicht:
399.36
Reinheit:
0.997
CAS Nummer:
[839712-25-3]
Formel:
C19H28Cl2N4O
Target-Kategorie:
Dopamine Receptor|||5-HT Receptor
T15117
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