Vactosertib Hydrochloride (EW-7197 Hydrochloride) is an orally active and highly efficient ATP-competitive ALK5 (activin receptor-like kinase 5) inhibitor, a TGF-beta receptor I inhibitor with anti-metastatic and anticancer properties. It sensitizes pancreatic cancer cells to gemcitabine by inhibiting their viability.
Molekulargewicht:
435.89
Reinheit:
0.9803
CAS Nummer:
[1352610-25-3]
Formel:
C22H19ClFN7
Target-Kategorie:
ALK|||TGF-beta/Smad
T15262
T15262
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