OP-3633 is an effective and selective steroidal glucocorticoid receptor (GR) antagonist (IC50: 29 nM). OP-3633 shows low progesterone receptor (PR) agonism and androgen receptor (AR) antagonism. It also has an inhibition of GR transcriptional activity.
Molekulargewicht:
445.64
CAS Nummer:
[2102494-14-2]
Formel:
C30H39NO2
Target-Kategorie:
Others|||Glucocorticoid Receptor
T16396
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