Opiranserin is a development as an injectable agent for the treatment of postoperative pain. Opiranserin is a non-opioid and non-NSAID analgesic candidate and is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A) (IC50s: 0.86 and 1.3 µM, respectively). Opiranserin displays antagonistic activity on rP2X3 (IC50=0.87 µM).
Molekulargewicht:
394.51
CAS Nummer:
[1441000-45-8]
Formel:
C21H34N2O5
Target-Kategorie:
GlyT|||5-HT Receptor|||P2X Receptor
T16399
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