YSY01A, CAS [[1194235-46-5]]

Artikelnummer: TGM-T200778
Artikelname: YSY01A, CAS [[1194235-46-5]]
Artikelnummer: TGM-T200778
Hersteller Artikelnummer: T200778
Alternativnummer: TGM-T200778-25MG,TGM-T200778-50MG,TGM-T200778-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
YSY01A is a proteasome inhibitor that suppresses cancer cell survival by inducing apoptosis (Apoptosis). It demonstrates IC50 values against various cell lines such as HEK293T, A549, MCF-7, MGC-803, and PC-3M with values of 51.01, 9.21, 5.21, 8.9, and 35.4 nM respectively. Additionally, YSY01A serves as a degrader of gp130 and JAK2, eliminating constitutive STAT3 signaling in human A549 lung cancer cells by downregulating gp130 and JAK2. YSY01A holds potential for research in cancer therapeutics.
Molekulargewicht: 547.45
CAS Nummer: [1194235-46-5]
Formel: C29H38BN5O5
Target-Kategorie: JAK|||Interleukin|||STAT|||Proteasome
T200778