PXS-4787 hydrochloride, CAS [[2409964-40-3]]

Artikelnummer: TGM-T201314
Artikelname: PXS-4787 hydrochloride, CAS [[2409964-40-3]]
Artikelnummer: TGM-T201314
Hersteller Artikelnummer: T201314
Alternativnummer: TGM-T201314-25MG,TGM-T201314-50MG,TGM-T201314-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
PXS-4787 hydrochloride is a specific and potent pan-lysyl oxidase inhibitor that effectively eliminates the activity of lysyl oxidase. It exhibits varying IC50 values against different forms of the enzyme, including 2 µM (Bovine LOX), 3.2 µM (rh LOXL1), 0.6 µM (rh LOXL2), 1.4 µM (rh LOXL3), and 0.2 µM (rh LOXL4). In addition, PXS-4787 hydrochloride reduces the deposition and cross-linking of collagen I secreted by human fibroblasts.
Molekulargewicht: 265.73
CAS Nummer: [2409964-40-3]
Formel: C10H13ClFNO2S
Target-Kategorie: Monoamine Oxidase
T201314