GP-515 HCl is an adenosine kinase inhibitor. In cultured rat myocardial myocytes (RMMs), GP-515 can induce the expression of vascular endothelial growth factor (VEGF). Under severe hypoxia (1% O(2)), GP-515 (20 microM) does not affect VEGF protein expression, but under mild hypoxic conditions, it increases VEGF expression by 27%.
Molekulargewicht:
345.15(free base)
CAS Nummer:
[144928-89-2]
Formel:
C10H13BrN6O3 xClH
T202308
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