PF-03654764 tosylate, CAS [[1337536-85-2]] Preis auf Anfrage

Artikelnummer: TGM-T202377
Artikelname: PF-03654764 tosylate, CAS [[1337536-85-2]] Preis auf Anfrage
Artikelnummer: TGM-T202377
Hersteller Artikelnummer: T202377
Alternativnummer: TGM-T202377-10MG,TGM-T202377-50MG
Hersteller: TargetMol
Kategorie: Biochemikalien
Alternative Synonym: OP970177FN , Q27285769
PF-03654764 exhibits high affinity for the human H3 receptor, but displays significantly lower affinity for the rat H3 receptor, with over 1000-fold selectivity against other human histamine receptor subtypes (H1, H2, and H4). In functional assays measuring cAMP using reporter gene assays (beta-lactamase) conducted in HEK293 cells stably expressing the full-length human or rat H3 receptor, PF-03654764 demonstrated potent antagonist properties.
CAS Nummer: [1337536-85-2]
Formel: C20H28F2N2O xC7H8O3S
T202377