MU1920 is an ATP-competitive, selective inhibitor of haspin with an IC50 of 6 nM. In mouse plasma and microsomes, it demonstrates favorable pharmacokinetic properties and metabolic stability. Although it lacks significant anticancer activity, MU1920 is suitable for developing chemical probes.
Molekulargewicht:
321.4
Formel:
C17H15N5S
Target-Kategorie:
Haspin Kinase
T204482
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