RSK2-IN-4 (Compound 10) is an inhibitor of RSK2, showing an inhibition rate of 13.73% on RSK2 activity at a concentration of 10 µM. It binds to the ATP binding site of RSK2 within the NTKD (N-terminal kinase domain), with the electron-donating group at the para position of the phenyl ring being crucial for its inhibitory activity.
Molekulargewicht:
258.706
CAS Nummer:
[62001-32-5]
Formel:
C13H11ClN4
Target-Kategorie:
S6 Kinase
T205512
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