BMY 7378 free base, CAS [[21102-94-3]] Preis auf Anfrage

Artikelnummer: TGM-T206148
Artikelname: BMY 7378 free base, CAS [[21102-94-3]] Preis auf Anfrage
Artikelnummer: TGM-T206148
Hersteller Artikelnummer: T206148
Alternativnummer: TGM-T206148-10MG,TGM-T206148-50MG
Hersteller: TargetMol
Kategorie: Biochemikalien
BMY 7378 (free base) is a selective antagonist for the alpha1D adrenergic receptor (alpha1D-AR). It exhibits a membrane-binding affinity for cloned rat alpha1D-AR (Ki=2 nM) that is over 100 times stronger than its affinity for cloned rat alpha1A-AR (Ki=800 nM) or hamster alpha1B-AR (Ki=600 nM). Additionally, BMY 7378 (free base) acts as a partial agonist at the 5-HT1A receptor.
Molekulargewicht: 385.5
CAS Nummer: [21102-94-3]
Formel: C22H31N3O3
Target-Kategorie: Adrenergic Receptor|||5-HT Receptor
T206148