BNS808 is an orally active, selective CB1R antagonist with an IC50 of 0.8 nM, demonstrating significant selectivity for CB2R and minimal brain penetration. It is being studied for the treatment of obesity and related metabolic complications, such as metabolic dysfunction-associated steatotic liver disease (MASLD). BNS808 reduces drug exposure to the central nervous system, enhancing safety, and minimizes drug interactions through high plasma protein binding.
Molekulargewicht:
548.869
CAS Nummer:
[2836313-12-1]
Formel:
C25H20Cl3N3O3S
Target-Kategorie:
Cannabinoid Receptor|||Cytochromes P450
T206797
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