uPSEM792 is a pharmacologically selective agonist molecule (PSEM) for PSAM4-GlyR, with an affinity Ki of 0.7 nM. It acts as a substrate for efflux transporters in both wild-type mice brains and in P-gp and BCRP double knockout mice. Additionally, uPSEM792 may serve as a lead compound in the development of PET radioligands for PSAM4-GlyR.
Molekulargewicht:
241.29
CAS Nummer:
[2323525-19-3]
Formel:
C14H15N3O
Target-Kategorie:
5-HT Receptor
T209079
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