Modzatinib, CAS [[2411407-25-3]]

Artikelnummer: TGM-T210785
Artikelname: Modzatinib, CAS [[2411407-25-3]]
Artikelnummer: TGM-T210785
Hersteller Artikelnummer: T210785
Alternativnummer: TGM-T210785-1MG, TGM-T210785-5MG, TGM-T210785-10MG
Hersteller: TargetMol
Kategorie: Biochemikalien
Alternative Synonym: ITK kinase-IN-1
Modzatinib (ITKkinase-IN-1) (compound I) is an inhibitor targeting ITK kinase with an IC50 of 8 nM in Jurkat cells, useful for researching inflammatory diseases. In hPBMC cells, it inhibits JAK3 with an IC50 of 23 nM (based on IL-2/pSTAT5 levels) and shows no inhibitory effect on JAK2.
Molekulargewicht: 361.39
Reinheit: 99.15%
CAS Nummer: [2411407-25-3]
Formel: C18H21F2N5O
Target-Kategorie: JAK|||Tyrosine Kinases