Modzatinib (ITKkinase-IN-1) (compound I) is an inhibitor targeting ITK kinase with an IC50 of 8 nM in Jurkat cells, useful for researching inflammatory diseases. In hPBMC cells, it inhibits JAK3 with an IC50 of 23 nM (based on IL-2/pSTAT5 levels) and shows no inhibitory effect on JAK2.
Molekulargewicht:
361.39
Reinheit:
99.15%
CAS Nummer:
[2411407-25-3]
Formel:
C18H21F2N5O
Target-Kategorie:
JAK|||Tyrosine Kinases
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