RGD-DA6 is an alphavbeta3-targeting ligand composed of RGDfK (an RGD peptide targeting integrin alphavbeta3), DOTADG, d-Glu, Lys, AMBA, and IPBA. Through radiolabeling, RGD-DA6 forms an alphavbeta3-targeted radioligand for high-contrast tumor imaging and improved anticancer efficacy.
Target-Kategorie:
Integrin
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