Bavdegalutamide (ARV-110) is an oral protein degrader that specifically binds to AR and mediates its degradation. Bavdegalutamide can degrade clinically relevant mutant AR proteins, maintain activity in a high androgen environment, and has an acceptable safety profile.
Molekulargewicht:
812.29
Reinheit:
99.96%
CAS Nummer:
[2222112-77-6]
Formel:
C41H43ClFN9O6
Target-Kategorie:
Androgen Receptor|||PROTACs
T22263
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