TP003 is a novel non-selective GABAA receptor benzodiazepine site agonist with affinity for alpha1beta2gam2, alpha2beta3gam2, alpha3beta3gam2, alpha5beta2gam2, EC50 of 20.3, 10.6, 3.24, 5.64 nM, respectively. TP003 has antianxiety and partial anticonvulsant activity via the alpha2GABAA receptor.
Molekulargewicht:
407.39
Reinheit:
99.17%
CAS Nummer:
[628690-75-5]
Formel:
C23H16F3N3O
Target-Kategorie:
GABA Receptor
T23466
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