J-104871 (UNII-6137X5QNJF) is a novel farnesyltransferase (FTase) inhibitor that competitively blocks Ras farnesylation in vivo, inhibits Ras processing in activated H-ras-transformed NIH3T3 cells, and suppresses tumor growth in nude mice transplanted with activated H-ras-transformed NIH3T3 cells.
Molekulargewicht:
708.67
Reinheit:
0.9903
CAS Nummer:
[191088-19-4]
Formel:
C38H32N2O12
Target-Kategorie:
Ras|||Transferase
T24188
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