Linifanib, CAS [[796967-16-3]]
Artikelnummer:
TGM-T2514
- Bilder (1)
| Artikelname: | Linifanib, CAS [[796967-16-3]] |
| Artikelnummer: | TGM-T2514 |
| Hersteller Artikelnummer: | T2514 |
| Alternativnummer: | TGM-T2514-1MLX10MM(INDMSO),TGM-T2514-5MG,TGM-T2514-10MG,TGM-T2514-25MG,TGM-T2514-50MG,TGM-T2514-100MG,TGM-T2514-200MG,TGM-T2514-500MG |
| Hersteller: | TargetMol |
| Kategorie: | Biochemikalien |
| Alternative Synonym: | ABT-869 , RG3635 , AL-39324 |
| Linifanib (AL-39324) (ABT-869) is a novel, potent ATP-competitive VEGFR/PDGFR inhibitor for KDR (IC50: 4 nM), CSF-1R (IC50: 3 nM), Flt-1/3 (IC50: 3/4 nM) and PDGFRbeta (IC50: 66 nM). Linifanib may exhibit potent antiproliferative and apoptotic effects on tumor cells whose proliferation is dependent on mutant kinases, such as FMS-related tyrosine kinase receptor-3 (FLT3). |
| Molekulargewicht: | 375.4 |
| Reinheit: | 98.00% |
| CAS Nummer: | [796967-16-3] |
| Formel: | C21H18FN5O |
| Target-Kategorie: | Apoptosis|||VEGFR|||FLT|||c-Fms|||CSF-1R|||Autophagy|||PDGFR|||c-Kit |

