NNC052090, CAS [[184845-43-0]]

Artikelnummer: TGM-T28183
Artikelname: NNC052090, CAS [[184845-43-0]]
Artikelnummer: TGM-T28183
Hersteller Artikelnummer: T28183
Alternativnummer: TGM-T28183-25MG,TGM-T28183-50MG,TGM-T28183-100MG
Hersteller: TargetMol
Kategorie: Biochemikalien
Alternative Synonym: NNC 052090 , NNC 05-2090 , NNC-052090 , NNC-05-2090 , NNC05-2090
NNC052090 is a GABA uptake inhibitor that displays moderate selectivity for BGT-1 transporters with Ki values are 1.4, 15, 19 and 41 µM for hBGT-1, hGAT-3, hGAT-1 and hGAT-2 respectively. NNC052090 also displays affinity at alpha1- and D2-receptors with IC50 values are 266 and 1632 nM respectively.
Molekulargewicht: 414.54
CAS Nummer: [184845-43-0]
Formel: C27H30N2O2
Target-Kategorie: Others|||GABA Receptor
T28183