A-366, CAS [[1527503-11-2]]

Produktübersicht

• Artikelname: A-366, CAS [[1527503-11-2]]
• Artikelnummer: TGM-T3624
• Hersteller Artikelnummer: T3624
• Alternativnummer: TGM-T3624-1MLX10MM(INDMSO),TGM-T3624-1MG,TGM-T3624-2MG,TGM-T3624-5MG,TGM-T3624-10MG,TGM-T3624-25MG,TGM-T3624-50MG,TGM-T3624-100MG
• Hersteller: TargetMol
• Kategorie: Biochemikalien
• Alternative Synonym: A 366 , A366

Produktbeschreibung

A-366 is a highly selective peptide-competitive histone methyltransferase G9a inhibitor with IC50s of 3.3 and 38 nM for G9a and GLP, respectively.It is more than 1,000-fold selective for G9a and GLP over the other 21 methyltransferases. It is an inhibitor of the Spindlin1-H3K4me3 interaction with an IC50 of 182.6 nM.It exhibits high affinity for human H3R with a Ki value of 17 nM, and shows subtype selectivity between subgroups of the histaminergic and dopaminergic receptor families.

Produkteigenschaften

• Molekulargewicht: 329.44
• Reinheit: 97.28%
• CAS Nummer: [1527503-11-2]
• Formel: C19H27N3O2
• Target-Kategorie: Histone Methyltransferase|||Epigenetic Reader Domain

Bilder

T3624