Relugolix, CAS [[737789-87-6]]

Artikelnummer: TGM-T3630
Artikelname: Relugolix, CAS [[737789-87-6]]
Artikelnummer: TGM-T3630
Hersteller Artikelnummer: T3630
Alternativnummer: TGM-T3630-1MLX10MM(INDMSO),TGM-T3630-2MG,TGM-T3630-5MG,TGM-T3630-10MG,TGM-T3630-25MG,TGM-T3630-50MG,TGM-T3630-100MG,TGM-T3630-200MG
Hersteller: TargetMol
Kategorie: Biochemikalien
Alternative Synonym: RVT-601 , TAK-385
Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, with potential antineoplastic activity. Relugolix competitively binds to and blocks the GnRH receptor in the anterior pituitary gland, which both prevents GnRH binding to the GnRH receptor and inhibits the secretion and release of both luteinizing hormone (LH) and follicle stimulating hormone (FSH). In males, the inhibition of LH secretion prevents the release of testosterone from Leydig cells in the testes. Since testosterone is required to sustain prostate growth, reducing testosterone levels may inhibit hormone-dependent prostate cancer cell proliferation.
Molekulargewicht: 623.63
Reinheit: 98.64%
CAS Nummer: [737789-87-6]
Formel: C29H27F2N7O5S
Target-Kategorie: GNRH Receptor
T3630