YNT-185 dihydrochloride, CAS [[1804978-82-2]]

Artikelnummer: TGM-T37112
Artikelname: YNT-185 dihydrochloride, CAS [[1804978-82-2]]
Artikelnummer: TGM-T37112
Hersteller Artikelnummer: T37112
Alternativnummer: TGM-T37112-2MG
Hersteller: TargetMol
Kategorie: Biochemikalien
Potent and selective orexin OX2 receptor agonist (EC50 = 28 nM at human OX2 expressed in CHO cells). Displays approximately 100-fold selectivity for OX2 over OX1 (EC50 = 2.75 µM at human OX1 expressed in CHO cells). Depolarizes OX2-expressing histaminergic neurons in mouse brain slices. Increases wake time in wild type mice. Suppresses cataplexy-like symptoms in OX knockout mice.
Molekulargewicht: 688.67
CAS Nummer: [1804978-82-2]
Formel: C33H39Cl2N5O5S
Target-Kategorie: Others|||OX Receptor
T37112