Bilaid C is a tetrapeptide µ-opioid receptor agonist (Ki= 210 nM in HEK293 cell membranes expressing the human receptor) that has been found inPenicillium.1It inhibits forskolin-induced cAMP accumulation by 77% in HEK293 cells expressing the human µ-opioid receptor when used at a concentration of 10 µM. Bilaid C induces inward rectifying potassium channel (Kir) currents in rat locus coeruleus slices that endogenously express high levels of the µ-opioid receptor (EC50= 4.2 µM).
Molekulargewicht:
526.62
CAS Nummer:
[2393866-13-0]
Formel:
C28H38N4O6
Target-Kategorie:
Opioid Receptor
T37199
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